9-hydroxy risperidone

It’s an active metabolite of risperidone. Risperidone is an atypical antipsychotic used to treat schizophrenia and bipolar disorder. It is an antagonist of the D1 as well as the D2 family receptors, and also against serotonin receptors.

By |2021-10-29T10:51:33+01:00October 29th, 2021|Comments Off on 9-hydroxy risperidone

Hydroxy itraconazole

It’s a metabolite of Itraconazole, an orally active antimycotic structurally related to Ketoconazole. It inhibits the fungal-mediated synthesis of ergosterol, via inhibition of lanosterol 14α-demethylase.

By |2021-10-29T10:47:34+01:00October 29th, 2021|Comments Off on Hydroxy itraconazole

4-Hydroxy nimesulide

It’s a biologically active metabolite of nimesulide. Nimesulide is a nonsteroidal anti-inflammatory drug (NSAID) used to treat pain and inflammatory diseases. NSAIDs work by inhibiting the activity of cyclooxygenase enzymes involved in the synthesis of key biological mediators, namely prostaglandins and thromboxanes.

By |2021-10-29T10:44:06+01:00October 29th, 2021|Comments Off on 4-Hydroxy nimesulide

4-Hydroxy Diclofenac

4Diclofenac is a nonsteroidal anti-inflammatory drug (NSAID) used to treat pain and inflammatory diseases. NSAIDs work by inhibiting the activity of cyclooxygenase enzymes involved in the synthesis of key biological mediators, namely prostaglandins and thromboxanes.

By |2021-10-29T10:40:36+01:00October 29th, 2021|Comments Off on 4-Hydroxy Diclofenac

4-hydroxyphenyl carvedilol

Carvedilol is both a non-selective β-adrenergic receptor antagonist (β1, β2) and an α-adrenergic receptor antagonist (α1). It is indicated in the management of high blood pressure and congestive heart failure (CHF).

By |2021-10-29T09:35:20+01:00October 19th, 2021|Comments Off on 4-hydroxyphenyl carvedilol

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